← Pipeline|Zenotinib

Zenotinib

Phase 2/3
451-1882
Source: Trial-derived·Trials: 1
Modality
Bispecific Ab
MOA
CD3xCD20
Target
PD-L1
Pathway
Angiogenesis
PNHMDS
Development Pipeline
Preclinical
~Jan 2019
~Apr 2020
Phase 1
~Jul 2020
~Oct 2021
Phase 2
Jan 2022
Apr 2031
Phase 2Current
NCT08330274
1,338 pts·MDS
2022-012031-04·Completed
1,338 total pts1 indication
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2031-04-025.0y awayPh3 Readout· MDS
Trial Timeline
2022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2
P2/3
Complet…
Catalysts
Ph3 Readout
2031-04-02 · 5.0y away
MDS
Completed|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT08330274Phase 2/3MDSCompleted1338BodyWt
Competitors (10)
DrugCompanyPhaseTargetMOA
LLY-1184Eli LillyNDA/BLAC5CD3xCD20
ZanuderotideNovartisPhase 1/2VEGFCD3xCD20
ABB-7516AbbViePhase 3PD-L1HPK1i
NVO-1361Novo NordiskPhase 3CD38CD3xCD20
ZorizanubrutinibNovo NordiskPhase 1BTKCD3xCD20
OlpatinibGSKPreclinicalPD-L1BCMA ADC
BAY-3684BayerApprovedPD-L1PARPi
PexamavacamtenDaiichi SankyoNDA/BLATIGITCD3xCD20
ITC-1028Intra-CellularPhase 2BCMACD3xCD20
PolatuximabNuvalentApprovedPD-L1PD-L1i