← Pipeline|Tixatapinarof

Tixatapinarof

Approved
RXR-6874
Source: Trial-derived·Trials: 3
Modality
Radioligand
MOA
BCMA ADC
Target
FGFR
Pathway
Notch
Asthma
Development Pipeline
Preclinical
~Nov 2009
~Feb 2011
Phase 1
~May 2011
~Aug 2012
Phase 2
~Nov 2012
~Feb 2014
Phase 3
~May 2014
~Aug 2015
NDA/BLA
~Nov 2015
~Feb 2017
Approved
May 2017
May 2031
ApprovedCurrent
NCT04085450
1,943 pts·Asthma
2020-082031-05·Recruiting
NCT07650272
2,979 pts·Asthma
2025-06TBD·Not yet recruiting
NCT04844680
1,079 pts·Asthma
2017-052030-07·Completed
6,001 total pts1 indication
CompletedCurrentUpcoming
Catalysts (2)
2030-07-224.3y awayPh3 Readout· Asthma
2031-05-035.1y awayPh3 Readout· Asthma
Trial Timeline
Q2Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2Q3
Approved
Complet…
Approved
Recruit…
Approved
Not yet…
Catalysts
Ph3 Readout
2030-07-22 · 4.3y away
Asthma
Ph3 Readout
2031-05-03 · 5.1y away
Asthma
RecruitingCompletedNot yet recruiting|StartCompletionToday
Trials (3)
NCTPhaseIndicationStatusNEP
NCT04085450ApprovedAsthmaRecruiting19436MWD
NCT07650272ApprovedAsthmaNot yet recr...2979UPCR
NCT04844680ApprovedAsthmaCompleted1079UPDRS
Competitors (10)
DrugCompanyPhaseTargetMOA
LLY-1592Eli LillyNDA/BLAFGFRBETi
DoxarasimodMerck & CoNDA/BLAFGFRKRASG12Di
AZN-3724AstraZenecaPreclinicalPSMABCMA ADC
AZN-7403AstraZenecaPhase 2/3FGFRTNFi
OlpatinibGSKPreclinicalPD-L1BCMA ADC
GIL-9779Gilead SciencesPhase 1IL-17ABCMA ADC
CevitinibRegeneronPhase 3FGFRPCSK9i
SematenlimabSamsung BiologicsPhase 3PI3KαBCMA ADC
TerazumabRecursionPhase 3AHRBCMA ADC
ABS-5770AbsciPreclinicalFGFRTROP-2 ADC