← Pipeline|Olpafutibatinib

Olpafutibatinib

Approved
IMC-6193
Source: Trial-derived·Trials: 4
Modality
Peptide
MOA
Menini
Target
SMN2
Pathway
RNA Splicing
NMOSDMigraine
Development Pipeline
Preclinical
~May 2011
~Aug 2012
Phase 1
~Nov 2012
~Feb 2014
Phase 2
~May 2014
~Aug 2015
Phase 3
~Nov 2015
~Feb 2017
NDA/BLA
~May 2017
~Aug 2018
Approved
Nov 2018
Oct 2031
ApprovedCurrent
NCT07515052
495 pts·NMOSD
2018-112031-05·Terminated
NCT06053301
1,089 pts·Migraine
2021-042031-10·Completed
NCT07306383
331 pts·Migraine
2023-122030-10·Recruiting
+1 more trial
3,319 total pts2 indications
CompletedCurrentUpcoming
Catalysts (3)
2030-10-274.6y awayPh3 Readout· Migraine
2031-05-055.1y awayPh3 Readout· NMOSD
2031-10-115.5y awayPh3 Readout· Migraine
Trial Timeline
Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2Q3Q4
Approved
Termina…
Approved
Complet…
Approved
Active
Approved
Recruit…
Catalysts
Ph3 Readout
2030-10-27 · 4.6y away
Migraine
Ph3 Readout
2031-05-05 · 5.1y away
NMOSD
Ph3 Readout
2031-10-11 · 5.5y away
Migraine
RecruitingActiveCompletedTerminated|StartCompletionToday
Trials (4)
NCTPhaseIndicationStatusNEP
NCT07515052ApprovedNMOSDTerminated495ACR20
NCT06053301ApprovedMigraineCompleted1089Safety
NCT07306383ApprovedMigraineRecruiting331LiverFat
NCT08360312ApprovedNMOSDActive1404UPCR
Competitors (10)
DrugCompanyPhaseTargetMOA
MavutenlimabJohnson & JohnsonPhase 3Cl18.2Menini
IvorelsinEli LillyApprovedJAK1Menini
NVO-2974Novo NordiskNDA/BLAPARPMenini
NVO-6275Novo NordiskPhase 1SMN2BTKi
TAK-5300TakedaPhase 1SMN2AuroraAi
GIL-2259Gilead SciencesApprovedSMN2CAR-T CD19
REG-647RegeneronPreclinicalSMN2SOS1i
TXG-675510x GenomicsApprovedCD123Menini
ZoricapivasertibCSL LimitedPhase 2HER2Menini
FixatapinarofJiangsu HengruiPreclinicalPLK4Menini