← Pipeline|Zenotapinarof

Zenotapinarof

Preclinical
VRT-4282
Source: Trial-derived·Trials: 1
Modality
Gene Therapy
MOA
IL-23i
Target
CD38
Pathway
T-cell
Cholangiocarcinoma
Development Pipeline
Preclinical
Dec 2024
Jun 2026
PreclinicalCurrent
NCT08329761
2,461 pts·Cholangiocarcinoma
2024-122026-06·Not yet recruiting
2,461 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2026-06-233mo awayInterim· Cholangiocarcinoma
Trial Timeline
2025Q2Q3Q42026Q2Q3
Preclinical
Not yet…
Catalysts
Interim
2026-06-23 · 3mo away
Cholangiocarcinoma
Not yet recruiting|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT08329761PreclinicalCholangiocarcinomaNot yet recr...2461CR
Competitors (10)
DrugCompanyPhaseTargetMOA
TerafutibatinibPfizerPhase 1/2CD38CGRPant
TirafotisoranRochePhase 2CD38CDK2i
NVS-6360NovartisApprovedCD38FXIai
DoxasotorasibAbbViePhase 2CD38VEGFi
SNY-2289SanofiPhase 2/3CD38IL-17i
NVO-1361Novo NordiskPhase 3CD38CD3xCD20
GSK-6983GSKPhase 2ALKIL-23i
MotarapivirGSKPreclinicalAuroraAIL-23i
AMG-2597AmgenPhase 2/3CD38PLK4i
IvosotorasibVertex PharmaPreclinicalCD38BTKi