← Pipeline|Elrarapivir

Elrarapivir

NDA/BLA
VRT-3718
Source: Trial-derived·Trials: 2
Modality
Vaccine
MOA
IL-17i
Target
PRMT5
Pathway
JAK/STAT
Rett
Development Pipeline
Preclinical
~Mar 2013
~Jun 2014
Phase 1
~Sep 2014
~Dec 2015
Phase 2
~Mar 2016
~Jun 2017
Phase 3
~Sep 2017
~Dec 2018
NDA/BLA
Mar 2019
Jan 2030
NDA/BLACurrent
NCT07306036
2,162 pts·Rett
2019-032029-04·Completed
NCT07966612
654 pts·Rett
2020-092030-01·Active
2,816 total pts1 indication
Approved
CompletedCurrentUpcoming
Catalysts (2)
2029-04-233.1y awayPh3 Readout· Rett
2030-01-183.8y awayPh3 Readout· Rett
Trial Timeline
2019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2
NDA/BLA
Complet…
NDA/BLA
Active
Catalysts
Ph3 Readout
2029-04-23 · 3.1y away
Rett
Ph3 Readout
2030-01-18 · 3.8y away
Rett
ActiveCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT07306036NDA/BLARettCompleted2162ORR
NCT07966612NDA/BLARettActive654MRD
Competitors (10)
DrugCompanyPhaseTargetMOA
NirarelsinJohnson & JohnsonPhase 2PRMT5CD47i
MRK-853Merck & CoPhase 1PRMT5WEE1i
GeliderotideSanofiPhase 1/2PRMT5JAK1i
SNY-2289SanofiPhase 2/3CD38IL-17i
CapifutibatinibSanofiApprovedPRMT5PI3Ki
NVO-9615Novo NordiskPhase 2/3PRMT5EZH2i
SuracageneGSKPhase 3PRMT5FcRni
FixainavolisibTakedaPreclinicalCDK2IL-17i
DarafutibatinibBioNTechPreclinicalPRMT5CFTRmod
RimaglumideBiogenPhase 1/2BCL-2IL-17i