← Pipeline|Rilutapinarof

Rilutapinarof

Phase 1
NUE-6133
Source: Trial-derived·Trials: 2
Modality
Vaccine
MOA
BCL-2i
Target
MET
Pathway
RNA Splicing
Parkinson'sObesity
Development Pipeline
Preclinical
~Feb 2019
~May 2020
Phase 1
Aug 2020
Apr 2030
Phase 1Current
NCT03813810
2,266 pts·Obesity
2020-082029-11·Completed
NCT07471166
1,716 pts·Parkinson's
2024-112030-04·Terminated
3,982 total pts2 indications
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2029-11-133.6y awayInterim· Obesity
2030-04-154.0y awayInterim· Parkinson's
Trial Timeline
Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2
P1
Complet…
P1
Termina…
Catalysts
Interim
2029-11-13 · 3.6y away
Obesity
Interim
2030-04-15 · 4.0y away
Parkinson's
CompletedTerminated|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT03813810Phase 1ObesityCompleted2266DAS28
NCT07471166Phase 1Parkinson'sTerminated17166MWD
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-5501PfizerPhase 1BTKBCL-2i
RHH-3592RochePhase 1/2GIP-RBCL-2i
GeliderotideNovartisNDA/BLAIL-17ABCL-2i
SNY-5783SanofiPhase 1/2METSTINGag
TezecilimabTakedaNDA/BLATauBCL-2i
RimaosocimabAmgenPreclinicalFXIaBCL-2i
SotosacituzumabVertex PharmaPhase 1METTYK2i
CapifutibatinibIncytePhase 3PCSK9BCL-2i
NBI-408NeurocrinePhase 2/3KRASG12DBCL-2i
HAL-996HalozymePhase 1/2BCL-2BCL-2i