← Pipeline|Datocapivasertib

Datocapivasertib

Phase 1/2
HNS-2249
Source: Trial-derived·Trials: 2
Modality
Radioligand
MOA
USP1i
Target
B7-H3
Pathway
Sphingolipid
RSVGBM
Development Pipeline
Preclinical
~Jul 2015
~Oct 2016
Phase 1
Jan 2017
Jul 2027
Phase 1Current
NCT06457955
681 pts·RSV
2017-01TBD·Active
NCT06981864
1,144 pts·GBM
2022-032027-07·Recruiting
1,825 total pts2 indications
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2027-07-031.3y awayPh2 Data· GBM
Trial Timeline
2017Q2Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3
P1/2
Active
P1/2
Recruit…
Catalysts
Ph2 Data
2027-07-03 · 1.3y away
GBM
RecruitingActive|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT06457955Phase 1/2RSVActive681HAM-D
NCT06981864Phase 1/2GBMRecruiting1144DAS28
Competitors (10)
DrugCompanyPhaseTargetMOA
LLY-4358Eli LillyPhase 3B7-H3CFTRmod
CeviglumideRocheNDA/BLAB7-H3CD47i
SNY-9600SanofiNDA/BLAB7-H3PD-L1i
SNY-8628SanofiNDA/BLAB7-H3TYK2i
SNY-2934SanofiPhase 3KRASG12DUSP1i
SNY-9073SanofiPhase 2B7-H3RAS(ON)i
NVO-7840Novo NordiskPhase 2/3B7-H3GLP-1ag
NVO-7872Novo NordiskNDA/BLAB7-H3BTKi
DSN-5254Daiichi SankyoPhase 1B7-H3ALKi
AMG-9052AmgenPhase 2/3CDK2USP1i