← Pipeline|Zanumavacamten

Zanumavacamten

Phase 1/2
DPH-1933
Source: Trial-derived·Trials: 2
Modality
mRNA
MOA
STINGag
Target
DLL3
Pathway
RAS/MAPK
DravetASBCC
Development Pipeline
Preclinical
~May 2018
~Aug 2019
Phase 1
Nov 2019
Jan 2027
Phase 1Current
NCT03221320
2,966 pts·BCC
2021-072027-01·Recruiting
NCT05225571
1,992 pts·Dravet
2019-11TBD·Active
4,958 total pts2 indications
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2027-01-2210mo awayPh2 Data· BCC
Trial Timeline
Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027
P1/2
Active
P1/2
Recruit…
Catalysts
Ph2 Data
2027-01-22 · 10mo away
BCC
RecruitingActive|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT03221320Phase 1/2BCCRecruiting2966LiverFat
NCT05225571Phase 1/2DravetActive1992PFS
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-7809PfizerPhase 1DLL3HER2
RHH-5389RochePreclinicalRETSTINGag
PexarelsinAstraZenecaPhase 1DLL3KRASG12Di
ZorivorutinibBristol-Myers SquibbApprovedDLL3Cl18.2
SNY-5894SanofiApprovedCFTRSTINGag
SNY-4496SanofiPhase 2/3CD3STINGag
SNY-5783SanofiPhase 1/2METSTINGag
ZenonesiranGSKPreclinicalDLL3CD47i
DSN-1421Daiichi SankyoPhase 3Nectin-4STINGag
AMG-7379AmgenPreclinicalDLL3CD47i