← Pipeline|Bemazanubrutinib

Bemazanubrutinib

Approved
DPH-168
Source: Trial-derived·Trials: 2
Modality
ERT
MOA
BCL-2i
Target
AuroraA
Pathway
Epigenetic
WilmsMDD
Development Pipeline
Preclinical
~Dec 2012
~Mar 2014
Phase 1
~Jun 2014
~Sep 2015
Phase 2
~Dec 2015
~Mar 2017
Phase 3
~Jun 2017
~Sep 2018
NDA/BLA
~Dec 2018
~Mar 2020
Approved
Jun 2020
Feb 2026
ApprovedCurrent
NCT04827012
2,841 pts·MDD
2025-032026-02·Completed
NCT06511071
448 pts·Wilms
2020-06TBD·Active
3,289 total pts2 indications
CompletedCurrentUpcoming
Catalysts (1)
2026-02-092mo agoPh3 Readout· MDD
Trial Timeline
Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026
Approved
Active
Approved
Complet…
Catalysts
Ph3 Readout
2026-02-09 · 2mo ago
MDD
ActiveCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT04827012ApprovedMDDCompleted2841Mayo
NCT06511071ApprovedWilmsActive448BodyWt
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-5501PfizerPhase 1BTKBCL-2i
RHH-3592RochePhase 1/2GIP-RBCL-2i
GeliderotideNovartisNDA/BLAIL-17ABCL-2i
MotarapivirGSKPreclinicalAuroraAIL-23i
TezecilimabTakedaNDA/BLATauBCL-2i
BAY-8733BayerPreclinicalAuroraABETi
RimaosocimabAmgenPreclinicalFXIaBCL-2i
BNT-8090BioNTechPhase 2AuroraAPD-L1i
ARG-6988ArgenxPreclinicalAuroraACDK2i
CapifutibatinibIncytePhase 3PCSK9BCL-2i