← Pipeline|Zenosertib

Zenosertib

Phase 2/3
RNA-1959
Source: Trial-derived·Trials: 1
Modality
ADC
MOA
PCSK9i
Target
FXIa
Pathway
T-cell
CTCLFabryHS
Development Pipeline
Preclinical
~Jan 2017
~Apr 2018
Phase 1
~Jul 2018
~Oct 2019
Phase 2
Jan 2020
Aug 2027
Phase 2Current
NCT03393431
2,361 pts·CTCL
2020-012027-08·Recruiting
2,361 total pts1 indication
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2026-09-236mo awayEnrollment Complete· CTCL
2027-08-151.4y awayPh3 Readout· CTCL
Trial Timeline
2020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q4
P2/3
Recruit…
Catalysts
Enrollment Complete
2026-09-23 · 6mo away
CTCL
Ph3 Readout
2027-08-15 · 1.4y away
CTCL
Recruiting|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT03393431Phase 2/3CTCLRecruiting2361LiverFat
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-1085PfizerPreclinicalFXIaPD-L1i
RHH-682RochePhase 2FXIaPRMT5i
RHH-7975RochePhase 3FXIaIL-13i
GozelemzoparlimabMerck & CoPhase 2FXIaKRASG12Ci
MRK-8368Merck & CoPhase 3ALKPCSK9i
RibofutibatinibAstraZenecaPhase 2/3SOS1PCSK9i
AZN-4015AstraZenecaPreclinicalBCMAPCSK9i
PexazasiranSanofiPreclinicalFXIaKRASG12Ci
PolazasiranAmgenPhase 2LAG-3PCSK9i
RimaosocimabAmgenPreclinicalFXIaBCL-2i