← Pipeline|Lirazanubrutinib

Lirazanubrutinib

Phase 1
532-2445
Source: Trial-derived·Trials: 2
Modality
Cell Therapy
MOA
Menini
Target
USP1
Pathway
Cell Cycle
PTSD
Development Pipeline
Preclinical
~May 2016
~Aug 2017
Phase 1
Nov 2017
Sep 2027
Phase 1Current
NCT06223259
2,833 pts·PTSD
2017-112026-07·Active
NCT08380557
943 pts·PTSD
2022-032027-09·Completed
3,776 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2026-07-224mo awayInterim· PTSD
2027-09-181.5y awayInterim· PTSD
Trial Timeline
Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q4
P1
Active
P1
Complet…
Catalysts
Interim
2026-07-22 · 4mo away
PTSD
Interim
2027-09-18 · 1.5y away
PTSD
ActiveCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT06223259Phase 1PTSDActive2833UPCR
NCT08380557Phase 1PTSDCompleted943ORR
Competitors (10)
DrugCompanyPhaseTargetMOA
MavutenlimabJohnson & JohnsonPhase 3Cl18.2Menini
IvorelsinEli LillyApprovedJAK1Menini
ABB-2476AbbViePhase 1/2USP1FcRni
NVO-2974Novo NordiskNDA/BLAPARPMenini
OlpafutibatinibImmunocoreApprovedSMN2Menini
TezesotorasibEnlivenPhase 2USP1MALT1i
ETN-506389bioPhase 1/2USP1Anti-Tau
TXG-675510x GenomicsApprovedCD123Menini
ZoricapivasertibCSL LimitedPhase 2HER2Menini
FixatapinarofJiangsu HengruiPreclinicalPLK4Menini