← Pipeline|Tiravorutinib

Tiravorutinib

Preclinical
MEI-2255
Source: Trial-derived·Trials: 1
Modality
Peptide
MOA
TNFi
Target
GLP-1R
Pathway
Hedgehog
CRCGastric Ca
Development Pipeline
Preclinical
Aug 2023
May 2025
PreclinicalCurrent
NCT04714580
1,572 pts·Gastric Ca
2023-082025-05·Active
1,572 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2025-05-2110mo agoInterim· Gastric Ca
Trial Timeline
Q42024Q2Q3Q42025Q2
Preclinical
Active
Catalysts
Interim
2025-05-21 · 10mo ago
Gastric Ca
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT04714580PreclinicalGastric CaActive1572eGFR
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-2191PfizerNDA/BLAGLP-1RSHP2i
RiboinavolisibJohnson & JohnsonPhase 2/3GLP-1RMALT1i
TirzepatideEli LillyApprovedGLP-1RGLP-1/GIP Dual Agonist
MRK-5413Merck & CoPhase 1GLP-1RVEGFi
AZN-7403AstraZenecaPhase 2/3FGFRTNFi
VoxacilimabAstraZenecaPhase 1/2GLP-1RPI3Ki
AZN-5171AstraZenecaApprovedGLP-1RGLP-1/GIP
TAK-8262TakedaNDA/BLATauTNFi
MavuglumideBayerApprovedGLP-1RCDK2i
BemarelsinDaiichi SankyoPreclinicalGLP-1RBiTE