← Pipeline|Tirazanubrutinib

Tirazanubrutinib

NDA/BLA
CYM-2367
Source: Trial-derived·Trials: 2
Modality
mAb
MOA
MALT1i
Target
MET
Pathway
NF-κB
SchizophreniaNBALL
Development Pipeline
Preclinical
~May 2017
~Aug 2018
Phase 1
~Nov 2018
~Feb 2020
Phase 2
~May 2020
~Aug 2021
Phase 3
~Nov 2021
~Feb 2023
NDA/BLA
May 2023
Jul 2029
NDA/BLACurrent
NCT05513828
962 pts·NB
2025-062029-07·Terminated
NCT04606982
1,217 pts·NB
2023-05TBD·Terminated
2,179 total pts1 indication
Approved
CompletedCurrentUpcoming
Catalysts (1)
2029-07-073.3y awayPh3 Readout· NB
Trial Timeline
Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3
NDA/BLA
Termina…
NDA/BLA
Termina…
Catalysts
Ph3 Readout
2029-07-07 · 3.3y away
NB
Terminated|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT05513828NDA/BLANBTerminated962HAM-D
NCT04606982NDA/BLANBTerminated1217SRI-4
Competitors (10)
DrugCompanyPhaseTargetMOA
JNJ-2735Johnson & JohnsonPhase 2/3Cl18.2MALT1i
RiboinavolisibJohnson & JohnsonPhase 2/3GLP-1RMALT1i
RHH-974RochePreclinicalJAK1MALT1i
NVS-3297NovartisPreclinicalCDK2MALT1i
ABB-8985AbbViePhase 2CD20MALT1i
SNY-5783SanofiPhase 1/2METSTINGag
SotosacituzumabVertex PharmaPhase 1METTYK2i
SovarelsinAlnylamPhase 2/3LAG-3MALT1i
ITC-6153Intra-CellularPhase 3KRASG12CMALT1i
GelisertibSamsung BiologicsApprovedIL-23MALT1i