← Pipeline|PLR-1516

PLR-1516

Phase 1
Source: Trial-derived·Trials: 2
Modality
Small Molecule
MOA
IL-17i
Target
Cl18.2
Pathway
Notch
MDDMDS
Development Pipeline
Preclinical
~Apr 2018
~Jul 2019
Phase 1
Oct 2019
Aug 2027
Phase 1Current
NCT08461111
2,528 pts·MDD
2019-102025-01·Completed
NCT07148694
691 pts·MDD
2023-012027-08·Active
3,219 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2025-01-181.2y agoInterim· MDD
2027-08-211.4y awayInterim· MDD
Trial Timeline
Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q4
P1
Complet…
P1
Active
Catalysts
Interim
2025-01-18 · 1.2y ago
MDD
Interim
2027-08-21 · 1.4y away
MDD
ActiveCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT08461111Phase 1MDDCompleted2528UPCR
NCT07148694Phase 1MDDActive691DOR
Competitors (10)
DrugCompanyPhaseTargetMOA
MavutenlimabJohnson & JohnsonPhase 3Cl18.2Menini
JNJ-2735Johnson & JohnsonPhase 2/3Cl18.2MALT1i
RibosacituzumabRocheApprovedCl18.2KIF18Ai
AdagrazumabNovartisPhase 2/3Cl18.2EZH2i
ZorimavacamtenBristol-Myers SquibbPreclinicalCl18.2CDK4/6i
SNY-2289SanofiPhase 2/3CD38IL-17i
FixainavolisibTakedaPreclinicalCDK2IL-17i
DoxafotisoranDaiichi SankyoPhase 1Cl18.2WEE1i
ElrarapivirVertex PharmaNDA/BLAPRMT5IL-17i
RimaglumideBiogenPhase 1/2BCL-2IL-17i