← Pipeline|Tirazanubrutinib

Tirazanubrutinib

Preclinical
PHA-1734
Source: Trial-derived·Trials: 2
Modality
mRNA
MOA
PD-L1i
Target
CDK2
Pathway
PI3K/AKT
SCLC
Development Pipeline
Preclinical
Aug 2019
Jul 2029
PreclinicalCurrent
NCT06970407
2,163 pts·SCLC
2019-082029-07·Recruiting
NCT06107366
1,386 pts·SCLC
2024-072028-01·Active
3,549 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2028-01-271.8y awayInterim· SCLC
2029-07-153.3y awayInterim· SCLC
Trial Timeline
Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3
Preclinical
Recruit…
Preclinical
Active
Catalysts
Interim
2028-01-27 · 1.8y away
SCLC
Interim
2029-07-15 · 3.3y away
SCLC
RecruitingActive|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT06970407PreclinicalSCLCRecruiting2163PANSS
NCT06107366PreclinicalSCLCActive1386LiverFat
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-3703PfizerPhase 1/2CDK2CDK2i
PFE-1085PfizerPreclinicalFXIaPD-L1i
NVS-3297NovartisPreclinicalCDK2MALT1i
RilulemzoparlimabNovartisPhase 2/3KRASG12DPD-L1i
SNY-9600SanofiNDA/BLAB7-H3PD-L1i
FixainavolisibTakedaPreclinicalCDK2IL-17i
NirafutibatinibBayerPhase 2WRNPD-L1i
AMG-1919AmgenPhase 2/3CDK2IL-13i
MotainavolisibAmgenNDA/BLACD47PD-L1i
AMG-415AmgenPhase 1CDK2MDM2i