← Pipeline|Zorisertib

Zorisertib

Approved
BIO-873
Source: Trial-derived·Trials: 1
Modality
Cell Therapy
MOA
TNFi
Target
SHP2
Pathway
PD-1/PD-L1
RSVParkinson'sThymoma
Development Pipeline
Preclinical
~Dec 2016
~Mar 2018
Phase 1
~Jun 2018
~Sep 2019
Phase 2
~Dec 2019
~Mar 2021
Phase 3
~Jun 2021
~Sep 2022
NDA/BLA
~Dec 2022
~Mar 2024
Approved
Jun 2024
Mar 2029
ApprovedCurrent
NCT06071844
302 pts·Thymoma
2024-062029-03·Terminated
302 total pts1 indication
CompletedCurrentUpcoming
Catalysts (1)
2029-03-133.0y awayPh3 Readout· Thymoma
Trial Timeline
Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2
Approved
Termina…
Catalysts
Ph3 Readout
2029-03-13 · 3.0y away
Thymoma
Terminated|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT06071844ApprovedThymomaTerminated302FEV1
Competitors (10)
DrugCompanyPhaseTargetMOA
NVS-5126NovartisPhase 3SHP2PI3Ki
MRK-1380Merck & CoPreclinicalSHP2SOS1i
ABB-1817AbbViePhase 3SHP2WRNi
AZN-7403AstraZenecaPhase 2/3FGFRTNFi
AZN-8281AstraZenecaPhase 1SHP2BTKi
AZN-8478AstraZenecaNDA/BLASHP2KRASG12Ci
TAK-8262TakedaNDA/BLATauTNFi
TalalemzoparlimabGilead SciencesPhase 1FcRnTNFi
MRN-7409ModernaNDA/BLASHP2CDK2i
RibozanubrutinibGenmabApprovedGPRC5DTNFi