← Pipeline|Capizanubrutinib

Capizanubrutinib

Preclinical
298-3597
Source: Trial-derived·Trials: 1
Modality
Bispecific Ab
MOA
FGFRi
Target
KRASG12C
Pathway
mTOR
Ewing SarcomaCervical Ca
Development Pipeline
Preclinical
Feb 2024
Dec 2030
PreclinicalCurrent
NCT08935535
2,320 pts·Ewing Sarcoma
2024-022030-12·Active
2,320 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2030-12-154.7y awayInterim· Ewing Sarcoma
Trial Timeline
2024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q4
Preclinical
Active
Catalysts
Interim
2030-12-15 · 4.7y away
Ewing Sarcoma
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT08935535PreclinicalEwing SarcomaActive2320ORR
Competitors (10)
DrugCompanyPhaseTargetMOA
JNJ-179Johnson & JohnsonApprovedKRASG12CBETi
LLY-9749Eli LillyPhase 3C5FGFRi
LLY-1956Eli LillyPhase 1/2BCMAFGFRi
BMY-4586Bristol-Myers SquibbPreclinicalKRASG12CIL-13i
DoxarapivirBristol-Myers SquibbPhase 3KRASG12CSOS1i
AMG-4531AmgenPhase 2/3KRASG12CPRMT5i
REG-8074RegeneronPhase 2/3KRASG12CCAR-T BCMA
VRT-1891Vertex PharmaPhase 1KRASG12CPRMT5i
PemitapinarofBeiGeneApprovedKRASG12CWRNi
SRP-9822SareptaPhase 3SOS1FGFRi