← Pipeline|GSK-2051

GSK-2051

Phase 1
By GSK
Source: Trial-derived·Trials: 2
Modality
Gene Editing
MOA
EGFRi
Target
PSMA
Pathway
Ferroptosis
Heart FailureDLBCLMigraine
Development Pipeline
Preclinical
~Sep 2017
~Dec 2018
Phase 1
Mar 2019
Jun 2027
Phase 1Current
NCT07702964
1,611 pts·Migraine
2019-032027-06·Not yet recruiting
NCT05469564
313 pts·DLBCL
2025-092025-10·Active
1,924 total pts2 indications
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2025-10-016mo agoInterim· DLBCL
2027-06-181.2y awayInterim· Migraine
Trial Timeline
2019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3
P1
Not yet…
P1
Active
Catalysts
Interim
2025-10-01 · 6mo ago
DLBCL
Interim
2027-06-18 · 1.2y away
Migraine
ActiveNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT07702964Phase 1MigraineNot yet recr...1611PASI75
NCT05469564Phase 1DLBCLActive313Safety
Competitors (10)
DrugCompanyPhaseTargetMOA
NiranesiranJohnson & JohnsonPhase 2KIF18AEGFRi
JNJ-5094Johnson & JohnsonPhase 2/3GIP-REGFRi
AZN-3724AstraZenecaPreclinicalPSMABCMA ADC
DoxacageneSanofiApprovedPSMASHP2i
GIL-2445Gilead SciencesPhase 2/3PSMAALKi
GIL-8529Gilead SciencesPhase 1/2JAK1EGFRi
BII-1564BiogenPhase 2PSMABETi
BGN-3859BeiGeneApprovedPSMACD47i
207-2754Samsung BiologicsPhase 1/2KRASG12DEGFRi
MavuratamabBlueprint MedicinesNDA/BLABETEGFRi