← Pipeline|Polatapinarof

Polatapinarof

Phase 1
255-5081
Source: Trial-derived·Trials: 1
Modality
siRNA
MOA
BCL-2i
Target
PRMT5
Pathway
Apoptosis
Schizophrenia
Development Pipeline
Preclinical
~May 2020
~Aug 2021
Phase 1
Nov 2021
Nov 2029
Phase 1Current
NCT08924117
2,998 pts·Schizophrenia
2021-112029-11·Not yet recruiting
2,998 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2029-11-043.6y awayInterim· Schizophrenia
Trial Timeline
Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q4
P1
Not yet…
Catalysts
Interim
2029-11-04 · 3.6y away
Schizophrenia
Not yet recruiting|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT08924117Phase 1SchizophreniaNot yet recr...2998Mayo
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-5501PfizerPhase 1BTKBCL-2i
NirarelsinJohnson & JohnsonPhase 2PRMT5CD47i
RHH-3592RochePhase 1/2GIP-RBCL-2i
GeliderotideNovartisNDA/BLAIL-17ABCL-2i
MRK-853Merck & CoPhase 1PRMT5WEE1i
GeliderotideSanofiPhase 1/2PRMT5JAK1i
CapifutibatinibSanofiApprovedPRMT5PI3Ki
NVO-9615Novo NordiskPhase 2/3PRMT5EZH2i
SuracageneGSKPhase 3PRMT5FcRni
TezecilimabTakedaNDA/BLATauBCL-2i