← Pipeline|Zenonesiran

Zenonesiran

Preclinical
GSK-4504
By GSK
Source: Trial-derived·Trials: 1
Modality
ADC
MOA
CD47i
Target
DLL3
Pathway
Checkpoint
DMDHemophilia A
Development Pipeline
Preclinical
Mar 2019
Mar 2030
PreclinicalCurrent
NCT04907615
126 pts·Hemophilia A
2019-032030-03·Completed
126 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2030-03-144.0y awayInterim· Hemophilia A
Trial Timeline
2019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2
Preclinical
Complet…
Catalysts
Interim
2030-03-14 · 4.0y away
Hemophilia A
Completed|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT04907615PreclinicalHemophilia ACompleted126MRD
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-7809PfizerPhase 1DLL3HER2
NirarelsinJohnson & JohnsonPhase 2PRMT5CD47i
CevizanubrutinibJohnson & JohnsonPreclinicalFcRnCD47i
CeviglumideRocheNDA/BLAB7-H3CD47i
NVS-1475NovartisPhase 2MeninCD47i
PexarelsinAstraZenecaPhase 1DLL3KRASG12Di
AZN-6294AstraZenecaPhase 2/3APOC3CD47i
ZorivorutinibBristol-Myers SquibbApprovedDLL3Cl18.2
AMG-7379AmgenPreclinicalDLL3CD47i
ARG-1924ArgenxPreclinicalDLL3JAK1i