← Pipeline|Doxasertib

Doxasertib

Preclinical
SYN-8630
Source: Trial-derived·Trials: 1
Modality
Radioligand
MOA
IL-23i
Target
AuroraA
Pathway
Autophagy
UCTTR Amyloidosis
Development Pipeline
Preclinical
Nov 2019
May 2028
PreclinicalCurrent
NCT06551124
766 pts·UC
2019-112028-05·Active
766 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2028-05-032.1y awayInterim· UC
Trial Timeline
Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3
Preclinical
Active
Catalysts
Interim
2028-05-03 · 2.1y away
UC
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT06551124PreclinicalUCActive766CfB
Competitors (10)
DrugCompanyPhaseTargetMOA
GSK-6983GSKPhase 2ALKIL-23i
MotarapivirGSKPreclinicalAuroraAIL-23i
BAY-8733BayerPreclinicalAuroraABETi
ZenotapinarofVertex PharmaPreclinicalCD38IL-23i
BNT-8090BioNTechPhase 2AuroraAPD-L1i
ARG-6988ArgenxPreclinicalAuroraACDK2i
BemasotorasibExelixisPhase 2CD38IL-23i
TirasotorasibViking TherapeuticsPhase 1CFTRIL-23i
SemamavacamtenIdeaya BioPhase 1/2AuroraABTKi
CevinaritidePraxis PrecisionPhase 3AuroraAFcRni