← Pipeline|Doxazanubrutinib

Doxazanubrutinib

Phase 3
PRO-5650
Source: Trial-derived·Trials: 1
Modality
Radioligand
MOA
Anti-Tau
Target
MALT1
Pathway
Hedgehog
FabryRCCPV
Development Pipeline
Preclinical
~Nov 2020
~Feb 2022
Phase 1
~May 2022
~Aug 2023
Phase 2
~Nov 2023
~Feb 2025
Phase 3
May 2025
Sep 2028
Phase 3Current
NCT03450065
2,306 pts·PV
2025-052028-09·Completed
2,306 total pts1 indication
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2028-09-262.5y awayPh3 Readout· PV
Trial Timeline
Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q4
P3
Complet…
Catalysts
Ph3 Readout
2028-09-26 · 2.5y away
PV
Completed|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT03450065Phase 3PVCompleted2306NT-proBNP
Competitors (10)
DrugCompanyPhaseTargetMOA
JNJ-8232Johnson & JohnsonNDA/BLAMALT1SGLT2i
RHH-7558RochePhase 1SGLT2Anti-Tau
NVS-5439NovartisPreclinicalBETAnti-Tau
BMY-7975Bristol-Myers SquibbPhase 1MALT1WRNi
NVO-9630Novo NordiskPhase 2CD3Anti-Tau
GSK-6516GSKPhase 1/2MALT1PARPi
REG-2172RegeneronPhase 1/2PCSK9Anti-Tau
BII-5240BiogenPhase 2/3MALT1HPK1i
ALN-3958AlnylamPhase 2MALT1PARPi
CevisacituzumabAlnylamPreclinicalMALT1SOS1i