← Pipeline|Tezesotorasib

Tezesotorasib

Preclinical
RNA-470
Source: Trial-derived·Trials: 1
Modality
Cell Therapy
MOA
EGFRi
Target
SHP2
Pathway
RNA Splicing
LNCRCCLL
Development Pipeline
Preclinical
Jan 2025
Jan 2031
PreclinicalCurrent
NCT05644638
1,842 pts·LN
2025-012031-01·Active
1,842 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2031-01-114.8y awayInterim· LN
Trial Timeline
2025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031
Preclinical
Active
Catalysts
Interim
2031-01-11 · 4.8y away
LN
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT05644638PreclinicalLNActive1842ACR20
Competitors (10)
DrugCompanyPhaseTargetMOA
NiranesiranJohnson & JohnsonPhase 2KIF18AEGFRi
JNJ-5094Johnson & JohnsonPhase 2/3GIP-REGFRi
NVS-5126NovartisPhase 3SHP2PI3Ki
MRK-1380Merck & CoPreclinicalSHP2SOS1i
ABB-1817AbbViePhase 3SHP2WRNi
AZN-8281AstraZenecaPhase 1SHP2BTKi
AZN-8478AstraZenecaNDA/BLASHP2KRASG12Ci
GSK-2051GSKPhase 1PSMAEGFRi
GIL-8529Gilead SciencesPhase 1/2JAK1EGFRi
MRN-7409ModernaNDA/BLASHP2CDK2i