← Pipeline|Tezezanubrutinib

Tezezanubrutinib

Preclinical
ATO-1130
Source: Trial-derived·Trials: 2
Modality
ERT
MOA
ALKi
Target
SHP2
Pathway
STING
PNHFLET
Development Pipeline
Preclinical
Nov 2017
Oct 2030
PreclinicalCurrent
NCT05687498
121 pts·PNH
2017-112030-10·Completed
NCT08033126
142 pts·FL
2024-11TBD·Recruiting
263 total pts2 indications
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2030-10-054.5y awayInterim· PNH
Trial Timeline
Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q4
Preclinical
Complet…
Preclinical
Recruit…
Catalysts
Interim
2030-10-05 · 4.5y away
PNH
RecruitingCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT05687498PreclinicalPNHCompleted121DOR
NCT08033126PreclinicalFLRecruiting142ACR20
Competitors (10)
DrugCompanyPhaseTargetMOA
MiriosocimabPfizerPhase 1PARPALKi
NVS-5126NovartisPhase 3SHP2PI3Ki
MRK-7739Merck & CoPreclinicalIL-23ALKi
MRK-1380Merck & CoPreclinicalSHP2SOS1i
ABB-1817AbbViePhase 3SHP2WRNi
AZN-8281AstraZenecaPhase 1SHP2BTKi
AZN-8478AstraZenecaNDA/BLASHP2KRASG12Ci
BMY-2495Bristol-Myers SquibbPhase 3KRASG12DALKi
DSN-5254Daiichi SankyoPhase 1B7-H3ALKi
SovacapivasertibAmgenPhase 3WEE1ALKi