← Pipeline|Tezevorutinib

Tezevorutinib

Approved
RNA-172
Source: Trial-derived·Trials: 1
Modality
Gene Editing
MOA
CD3xCD20
Target
SHP2
Pathway
Incretin
Angelman
Development Pipeline
Preclinical
~Mar 2010
~Jun 2011
Phase 1
~Sep 2011
~Dec 2012
Phase 2
~Mar 2013
~Jun 2014
Phase 3
~Sep 2014
~Dec 2015
NDA/BLA
~Mar 2016
~Jun 2017
Approved
Sep 2017
Jan 2028
ApprovedCurrent
NCT05096523
388 pts·Angelman
2017-092028-01·Completed
388 total pts1 indication
CompletedCurrentUpcoming
Catalysts (1)
2028-01-011.8y awayPh3 Readout· Angelman
Trial Timeline
Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028
Approved
Complet…
Catalysts
Ph3 Readout
2028-01-01 · 1.8y away
Angelman
Completed|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT05096523ApprovedAngelmanCompleted388DOR
Competitors (10)
DrugCompanyPhaseTargetMOA
LLY-1184Eli LillyNDA/BLAC5CD3xCD20
NVS-5126NovartisPhase 3SHP2PI3Ki
ZanuderotideNovartisPhase 1/2VEGFCD3xCD20
MRK-1380Merck & CoPreclinicalSHP2SOS1i
ABB-1817AbbViePhase 3SHP2WRNi
AZN-8281AstraZenecaPhase 1SHP2BTKi
AZN-8478AstraZenecaNDA/BLASHP2KRASG12Ci
NVO-1361Novo NordiskPhase 3CD38CD3xCD20
ZorizanubrutinibNovo NordiskPhase 1BTKCD3xCD20
PexamavacamtenDaiichi SankyoNDA/BLATIGITCD3xCD20