← Pipeline|Pexasertib

Pexasertib

Preclinical
ATL-9971
Source: Trial-derived·Trials: 2
Modality
Small Molecule
MOA
KIF18Ai
Target
CD38
Pathway
Incretin
NBFSGSGBM
Development Pipeline
Preclinical
Jun 2019
Jun 2031
PreclinicalCurrent
NCT03362083
2,943 pts·NB
2019-062031-06·Recruiting
NCT08444500
1,850 pts·GBM
2021-022028-10·Not yet recruiting
4,793 total pts2 indications
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2028-10-232.6y awayInterim· GBM
2031-06-115.2y awayInterim· NB
Trial Timeline
Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2Q3
Preclinical
Recruit…
Preclinical
Not yet…
Catalysts
Interim
2028-10-23 · 2.6y away
GBM
Interim
2031-06-11 · 5.2y away
NB
RecruitingNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT03362083PreclinicalNBRecruiting2943UPDRS
NCT08444500PreclinicalGBMNot yet recr...1850UPCR
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-7550PfizerPhase 3KIF18Ai
TerafutibatinibPfizerPhase 1/2CD38CGRPant
RibosacituzumabRocheApprovedCl18.2KIF18Ai
RHH-8482RochePhase 1BTKKIF18Ai
TirafotisoranRochePhase 2CD38CDK2i
PexatenlimabNovartisPhase 1/2GPRC5DKIF18Ai
NVS-6360NovartisApprovedCD38FXIai
DoxasotorasibAbbViePhase 2CD38VEGFi
SNY-2289SanofiPhase 2/3CD38IL-17i
NVO-1361Novo NordiskPhase 3CD38CD3xCD20