← Pipeline|Tirazanubrutinib

Tirazanubrutinib

Phase 1
FLA-2179
Source: Trial-derived·Trials: 1
Modality
Radioligand
MOA
HER2
Target
ALK
Pathway
JAK/STAT
RACKD
Development Pipeline
Preclinical
~Oct 2018
~Jan 2020
Phase 1
Apr 2020
Aug 2027
Phase 1Current
NCT05472272
23 pts·RA
2020-042027-08·Active
23 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2027-08-261.4y awayInterim· RA
Trial Timeline
Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q4
P1
Active
Catalysts
Interim
2027-08-26 · 1.4y away
RA
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT05472272Phase 1RAActive23PASI75
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-7809PfizerPhase 1DLL3HER2
LLY-8903Eli LillyPreclinicalCD47HER2
MRK-8368Merck & CoPhase 3ALKPCSK9i
SNY-7254SanofiPhase 2CFTRHER2
DatobrutinibSanofiPhase 3HER2
GSK-6983GSKPhase 2ALKIL-23i
TAK-9344TakedaPhase 3CGRPHER2
BAY-3308BayerPhase 1ALKSGLT2i
TixarelsinVertex PharmaPhase 1ALKRAS(ON)i
VRT-6833Vertex PharmaPreclinicalALKVEGFi