← Pipeline|ENT-2952

ENT-2952

Phase 3
Source: Trial-derived·Trials: 4
Modality
ERT
MOA
PARPi
Target
JAK2
Pathway
Wnt
CTCLThymoma
Development Pipeline
Preclinical
~Dec 2014
~Mar 2016
Phase 1
~Jun 2016
~Sep 2017
Phase 2
~Dec 2017
~Mar 2019
Phase 3
Jun 2019
May 2031
Phase 3Current
NCT07690229
2,994 pts·CTCL
2019-062025-04·Terminated
NCT03979891
2,869 pts·Thymoma
2020-082025-02·Active
NCT03128068
781 pts·Thymoma
2022-072030-09·Active
+1 more trial
8,621 total pts2 indications
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (4)
2025-02-191.1y agoPh3 Readout· Thymoma
2025-04-1412mo agoPh3 Readout· CTCL
2030-09-014.4y awayPh3 Readout· Thymoma
2031-05-255.1y awayPh3 Readout· CTCL
Trial Timeline
Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2Q3
P3
Termina…
P3
Active
P3
Active
P3
Termina…
Catalysts
Ph3 Readout
2025-02-19 · 1.1y ago
Thymoma
Ph3 Readout
2025-04-14 · 12mo ago
CTCL
Ph3 Readout
2030-09-01 · 4.4y away
Thymoma
Ph3 Readout
2031-05-25 · 5.1y away
CTCL
ActiveTerminated|StartCompletionToday
Trials (4)
NCTPhaseIndicationStatusNEP
NCT07690229Phase 3CTCLTerminated2994UPCR
NCT03979891Phase 3ThymomaActive2869HbA1c
NCT03128068Phase 3ThymomaActive7816MWD
NCT08235057Phase 3CTCLTerminated1977EDSS
Competitors (10)
DrugCompanyPhaseTargetMOA
MRK-3732Merck & CoPhase 1TYK2PARPi
GSK-6516GSKPhase 1/2MALT1PARPi
BAY-3684BayerApprovedPD-L1PARPi
BNT-5232BioNTechNDA/BLATIGITPARPi
ALN-3958AlnylamPhase 2MALT1PARPi
GMA-5010GenmabPhase 3JAK2TROP-2 ADC
CevifotisoranNeurocrineApprovedCD47PARPi
LEG-6533Legend BiotechNDA/BLAVEGFPARPi
LEG-9870Legend BiotechPhase 1CGRPPARPi
UTH-9370United TherapeuticsNDA/BLATIGITPARPi