← Pipeline|Pexarelsin

Pexarelsin

Phase 1
AZN-9004
Source: Trial-derived·Trials: 2
Modality
Cell Therapy
MOA
KRASG12Di
Target
DLL3
Pathway
RNA Splicing
CMLFL
Development Pipeline
Preclinical
~Mar 2016
~Jun 2017
Phase 1
Sep 2017
Aug 2028
Phase 1Current
NCT05618377
205 pts·FL
2017-092028-08·Not yet recruiting
NCT04703881
1,171 pts·FL
2024-08TBD·Terminated
1,376 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2028-08-012.3y awayInterim· FL
Trial Timeline
Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q4
P1
Not yet…
P1
Termina…
Catalysts
Interim
2028-08-01 · 2.3y away
FL
TerminatedNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT05618377Phase 1FLNot yet recr...205eGFR
NCT04703881Phase 1FLTerminated1171LiverFat
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-7809PfizerPhase 1DLL3HER2
DoxarasimodMerck & CoNDA/BLAFGFRKRASG12Di
ZanusertibAbbVieApprovedPCSK9KRASG12Di
ZorivorutinibBristol-Myers SquibbApprovedDLL3Cl18.2
ZenonesiranGSKPreclinicalDLL3CD47i
IvotuximabGSKNDA/BLAGIP-RKRASG12Di
AMG-7379AmgenPreclinicalDLL3CD47i
ARG-1924ArgenxPreclinicalDLL3JAK1i
CevinaritideGenmabPhase 2/3DLL3PD-1i
TerarasimodKrystal BiotechPhase 1/2PI3KαKRASG12Di