← Pipeline|Rimatinib

Rimatinib

NDA/BLA
BOU-2608
Source: Trial-derived·Trials: 2
Modality
Degrader
MOA
Anti-Tau
Target
VEGF
Pathway
Wnt
ADHDSCLC
Development Pipeline
Preclinical
~Jul 2011
~Oct 2012
Phase 1
~Jan 2013
~Apr 2014
Phase 2
~Jul 2014
~Oct 2015
Phase 3
~Jan 2016
~Apr 2017
NDA/BLA
Jul 2017
May 2026
NDA/BLACurrent
NCT05024244
120 pts·ADHD
2025-022025-10·Completed
NCT07256886
2,744 pts·ADHD
2017-072026-05·Not yet recruiting
2,864 total pts1 indication
Approved
CompletedCurrentUpcoming
Catalysts (2)
2025-10-076mo agoPh3 Readout· ADHD
2026-05-021mo awayPh3 Readout· ADHD
Trial Timeline
Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3
NDA/BLA
Not yet…
NDA/BLA
Complet…
Catalysts
Ph3 Readout
2025-10-07 · 6mo ago
ADHD
Ph3 Readout
2026-05-02 · 1mo away
ADHD
CompletedNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT05024244NDA/BLAADHDCompleted120ACR20
NCT07256886NDA/BLAADHDNot yet recr...2744PASI75
Competitors (10)
DrugCompanyPhaseTargetMOA
RHH-7558RochePhase 1SGLT2Anti-Tau
NVS-5439NovartisPreclinicalBETAnti-Tau
ZanuderotideNovartisPhase 1/2VEGFCD3xCD20
NVO-9630Novo NordiskPhase 2CD3Anti-Tau
TAK-8730TakedaPhase 2VEGFFXIai
GIL-2011Gilead SciencesPreclinicalVEGFSOS1i
BemazumabRegeneronPhase 1VEGFTROP-2 ADC
REG-2172RegeneronPhase 1/2PCSK9Anti-Tau
BGN-3305BeiGenePhase 2BCMAAnti-Tau
PemicapivasertibLegend BiotechPhase 3VEGFCDK4/6i