← Pipeline|Pexazanubrutinib

Pexazanubrutinib

Preclinical
OPT-2935
Source: Trial-derived·Trials: 1
Modality
mRNA
MOA
IL-17i
Target
TROP-2
Pathway
PI3K/AKT
MDSTTR AmyloidosisBladder Ca
Development Pipeline
Preclinical
Aug 2017
Jan 2026
PreclinicalCurrent
NCT07977542
1,479 pts·Bladder Ca
2017-082026-01·Active
1,479 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2026-01-182mo agoInterim· Bladder Ca
Trial Timeline
Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026
Preclinical
Active
Catalysts
Interim
2026-01-18 · 2mo ago
Bladder Ca
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT07977542PreclinicalBladder CaActive1479FEV1
Competitors (10)
DrugCompanyPhaseTargetMOA
NVS-4076NovartisPreclinicalTROP-2DLL3 ADC
NVS-8902NovartisPreclinicalTROP-2IL-13i
SNY-2289SanofiPhase 2/3CD38IL-17i
ZanumavacamtenGSKPhase 2/3TROP-2BTKi
FixainavolisibTakedaPreclinicalCDK2IL-17i
ElrarapivirVertex PharmaNDA/BLAPRMT5IL-17i
RimaglumideBiogenPhase 1/2BCL-2IL-17i
ARG-3458ArgenxPreclinicalRETIL-17i
ION-1378IonisNDA/BLATROP-2RAS(ON)i
NirafotisoranJazz PharmaPhase 2/3TROP-2SHP2i