← Pipeline|Tezesacituzumab

Tezesacituzumab

NDA/BLA
600-3446
Source: Trial-derived·Trials: 1
Modality
mAb
MOA
PRMT5i
Target
IL-23
Pathway
Epigenetic
CLLCeliac
Development Pipeline
Preclinical
~Mar 2012
~Jun 2013
Phase 1
~Sep 2013
~Dec 2014
Phase 2
~Mar 2015
~Jun 2016
Phase 3
~Sep 2016
~Dec 2017
NDA/BLA
Mar 2018
Aug 2025
NDA/BLACurrent
NCT08278559
1,494 pts·CLL
2018-032025-08·Recruiting
1,494 total pts1 indication
Approved
CompletedCurrentUpcoming
Catalysts (1)
2025-08-038mo agoPh3 Readout· CLL
Trial Timeline
Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3
NDA/BLA
Recruit…
Catalysts
Ph3 Readout
2025-08-03 · 8mo ago
CLL
Recruiting|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT08278559NDA/BLACLLRecruiting1494BodyWt
Competitors (10)
DrugCompanyPhaseTargetMOA
LLY-6079Eli LillyPhase 2MDM2PRMT5i
RHH-8550RocheApprovedBCL-2PRMT5i
RHH-682RochePhase 2FXIaPRMT5i
MRK-7739Merck & CoPreclinicalIL-23ALKi
TalainavolisibNovo NordiskPreclinicalKRASG12DPRMT5i
TerasacituzumabNovo NordiskNDA/BLAIL-23KRASG12Ci
DSN-6862Daiichi SankyoPreclinicalIL-23SOS1i
AMG-4531AmgenPhase 2/3KRASG12CPRMT5i
GIL-9142Gilead SciencesPhase 1FXIaPRMT5i
SemainavolisibGilead SciencesPhase 2PARPPRMT5i