← Pipeline|Voxabrutinib

Voxabrutinib

Phase 1/2
ANN-1950
Source: Trial-derived·Trials: 2
Modality
Vaccine
MOA
CGRPant
Target
EZH2
Pathway
PI3K/AKT
CMLTTR AmyloidosisNSCLC
Development Pipeline
Preclinical
~Mar 2021
~Jun 2022
Phase 1
Sep 2022
Sep 2028
Phase 1Current
NCT06682025
148 pts·NSCLC
2022-092025-01·Active
NCT04244914
1,392 pts·CML
2025-032028-09·Completed
1,540 total pts2 indications
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2025-01-101.2y agoPh2 Data· NSCLC
2028-09-032.4y awayPh2 Data· CML
Trial Timeline
Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q4
P1/2
Active
P1/2
Complet…
Catalysts
Ph2 Data
2025-01-10 · 1.2y ago
NSCLC
Ph2 Data
2028-09-03 · 2.4y away
CML
ActiveCompleted|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT06682025Phase 1/2NSCLCActive148BodyWt
NCT04244914Phase 1/2CMLCompleted1392ACR20
Competitors (10)
DrugCompanyPhaseTargetMOA
TerafutibatinibPfizerPhase 1/2CD38CGRPant
SotovorutinibPfizerApprovedCGRPant
ABB-3060AbbViePhase 2LAG-3CGRPant
DSN-2247Daiichi SankyoNDA/BLAEZH2C5i
GIL-6239Gilead SciencesPhase 2TNFαCGRPant
TezecilimabRegeneronApprovedIL-23CGRPant
INC-2432IncytePhase 2CD47CGRPant
SematapinarofLegend BiotechNDA/BLAVEGFCGRPant
HAL-9635HalozymePhase 2/3EZH2Cl18.2
RilufotisoranSamsung BiologicsNDA/BLAFXIaCGRPant