← Pipeline|Tezesotorasib

Tezesotorasib

Phase 2
ELV-9243
Source: Trial-derived·Trials: 2
Modality
ERT
MOA
MALT1i
Target
USP1
Pathway
Innate Imm
Atopic DermHSDravet
Development Pipeline
Preclinical
~Sep 2018
~Dec 2019
Phase 1
~Mar 2020
~Jun 2021
Phase 2
Sep 2021
Feb 2031
Phase 2Current
NCT04181919
2,685 pts·Dravet
2021-092031-02·Not yet recruiting
NCT03446148
112 pts·Dravet
2024-022030-10·Completed
2,797 total pts1 indication
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2030-10-184.6y awayPh2 Data· Dravet
2031-02-164.9y awayPh2 Data· Dravet
Trial Timeline
Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2
P2
Not yet…
P2
Complet…
Catalysts
Ph2 Data
2030-10-18 · 4.6y away
Dravet
Ph2 Data
2031-02-16 · 4.9y away
Dravet
CompletedNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT04181919Phase 2DravetNot yet recr...2685ORR
NCT03446148Phase 2DravetCompleted112EASI-75
Competitors (10)
DrugCompanyPhaseTargetMOA
JNJ-2735Johnson & JohnsonPhase 2/3Cl18.2MALT1i
RiboinavolisibJohnson & JohnsonPhase 2/3GLP-1RMALT1i
RHH-974RochePreclinicalJAK1MALT1i
NVS-3297NovartisPreclinicalCDK2MALT1i
ABB-2476AbbViePhase 1/2USP1FcRni
ABB-8985AbbViePhase 2CD20MALT1i
SovarelsinAlnylamPhase 2/3LAG-3MALT1i
ITC-6153Intra-CellularPhase 3KRASG12CMALT1i
GelisertibSamsung BiologicsApprovedIL-23MALT1i
RVM-7089Revolution MedicinesPhase 3IL-17AMALT1i