← Pipeline|Fixazanubrutinib

Fixazanubrutinib

Preclinical
ZTS-9957
Source: Trial-derived·Trials: 1
Modality
Gene Editing
MOA
USP1i
Target
EZH2
Pathway
Ferroptosis
AsthmaEwing SarcomaCervical Ca
Development Pipeline
Preclinical
May 2021
May 2030
PreclinicalCurrent
NCT08316834
2,266 pts·Ewing Sarcoma
2021-052030-05·Completed
2,266 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2030-05-034.1y awayInterim· Ewing Sarcoma
Trial Timeline
Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3
Preclinical
Complet…
Catalysts
Interim
2030-05-03 · 4.1y away
Ewing Sarcoma
Completed|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT08316834PreclinicalEwing SarcomaCompleted2266VA
Competitors (10)
DrugCompanyPhaseTargetMOA
SNY-2934SanofiPhase 3KRASG12DUSP1i
DSN-2247Daiichi SankyoNDA/BLAEZH2C5i
AMG-9052AmgenPhase 2/3CDK2USP1i
DatozumabRegeneronPhase 1B7-H3USP1i
GMA-729GenmabPhase 2BCL-2USP1i
HAL-9635HalozymePhase 2/3EZH2Cl18.2
PexanaritideInnovent BioPreclinicalSGLT2USP1i
ROI-9675Roivant SciencesNDA/BLAHER2USP1i
ITO-535iTeosNDA/BLAMDM2USP1i
TezeratamabPrime MedicinePhase 3CGRPUSP1i