← Pipeline|Darasertib

Darasertib

Phase 1/2
HEL-9266
Source: Trial-derived·Trials: 2
Modality
Cell Therapy
MOA
Menini
Target
PI3Kα
Pathway
RNA Splicing
SCDAtopic Derm
Development Pipeline
Preclinical
~Aug 2017
~Nov 2018
Phase 1
Feb 2019
Dec 2030
Phase 1Current
NCT04844513
1,351 pts·Atopic Derm
2022-032030-12·Not yet recruiting
NCT05030337
665 pts·SCD
2019-022025-09·Recruiting
2,016 total pts2 indications
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2025-09-216mo agoPh2 Data· SCD
2030-12-284.7y awayPh2 Data· Atopic Derm
Trial Timeline
2019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q4
P1/2
Recruit…
P1/2
Not yet…
Catalysts
Ph2 Data
2025-09-21 · 6mo ago
SCD
Ph2 Data
2030-12-28 · 4.7y away
Atopic Derm
RecruitingNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT04844513Phase 1/2Atopic DermNot yet recr...1351BodyWt
NCT05030337Phase 1/2SCDRecruiting665Biomarker
Competitors (10)
DrugCompanyPhaseTargetMOA
VoxaderotideJohnson & JohnsonNDA/BLAPI3KαIL-13i
MavutenlimabJohnson & JohnsonPhase 3Cl18.2Menini
IvorelsinEli LillyApprovedJAK1Menini
RimamavacamtenMerck & CoPhase 1PI3KαDLL3 ADC
NVO-2974Novo NordiskNDA/BLAPARPMenini
FixazanubrutinibAmgenPhase 2PI3KαCAR-T BCMA
GMA-1468GenmabNDA/BLAPI3KαWEE1i
369-789Hansoh PharmaPhase 3PI3KαTNFi
MavutuximabHansoh PharmaPhase 2/3PI3KαPCSK9i
SematenlimabSamsung BiologicsPhase 3PI3KαBCMA ADC