← Pipeline|Rimavorutinib

Rimavorutinib

Phase 3
THA-9471
Source: Trial-derived·Trials: 3
Modality
Small Molecule
MOA
CAR-T BCMA
Target
PARP
Pathway
Angiogenesis
ACCProstate CaCTCL
Development Pipeline
Preclinical
~Feb 2015
~May 2016
Phase 1
~Aug 2016
~Nov 2017
Phase 2
~Feb 2018
~May 2019
Phase 3
Aug 2019
Jul 2030
Phase 3Current
NCT04919990
2,676 pts·ACC
2019-082026-04·Active
NCT07127535
1,779 pts·CTCL
2021-122029-03·Completed
NCT05893622
500 pts·Prostate Ca
2020-052030-07·Terminated
4,955 total pts3 indications
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (3)
2026-04-112w awayPh3 Readout· ACC
2029-03-173.0y awayPh3 Readout· CTCL
2030-07-034.3y awayPh3 Readout· Prostate Ca
Trial Timeline
Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3
P3
Active
P3
Termina…
P3
Complet…
Catalysts
Ph3 Readout
2026-04-11 · 2w away
ACC
Ph3 Readout
2029-03-17 · 3.0y away
CTCL
Ph3 Readout
2030-07-03 · 4.3y away
Prostate Ca
ActiveCompletedTerminated|StartCompletionToday
Trials (3)
NCTPhaseIndicationStatusNEP
NCT04919990Phase 3ACCActive2676ACR20
NCT07127535Phase 3CTCLCompleted1779Mayo
NCT05893622Phase 3Prostate CaTerminated500HAM-D
Competitors (10)
DrugCompanyPhaseTargetMOA
MiriosocimabPfizerPhase 1PARPALKi
VoxacilimabPfizerPhase 2TYK2CAR-T BCMA
NVO-2974Novo NordiskNDA/BLAPARPMenini
NVO-9087Novo NordiskPhase 1/2TauCAR-T BCMA
FixazanubrutinibAmgenPhase 2PI3KαCAR-T BCMA
SemainavolisibGilead SciencesPhase 2PARPPRMT5i
REG-861RegeneronPhase 2PARPAuroraAi
REG-8074RegeneronPhase 2/3KRASG12CCAR-T BCMA
JAZ-8729Jazz PharmaPhase 2/3FcRnCAR-T BCMA
ACA-2691Acadia PharmaPhase 3BCMACAR-T BCMA