← Pipeline|Semazanubrutinib

Semazanubrutinib

Phase 3
NWR-247
Source: Trial-derived·Trials: 2
Modality
Radioligand
MOA
Anti-Tau
Target
TROP-2
Pathway
Tau
Parkinson'sCervical Ca
Development Pipeline
Preclinical
~Jul 2016
~Oct 2017
Phase 1
~Jan 2018
~Apr 2019
Phase 2
~Jul 2019
~Oct 2020
Phase 3
Jan 2021
Jun 2028
Phase 3Current
NCT07436063
2,541 pts·Parkinson's
2021-012028-06·Terminated
NCT03193125
1,190 pts·Cervical Ca
2022-012026-08·Completed
3,731 total pts2 indications
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2026-08-104mo awayPh3 Readout· Cervical Ca
2028-06-232.2y awayPh3 Readout· Parkinson's
Trial Timeline
2021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3
P3
Termina…
P3
Complet…
Catalysts
Ph3 Readout
2026-08-10 · 4mo away
Cervical Ca
Ph3 Readout
2028-06-23 · 2.2y away
Parkinson's
CompletedTerminated|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT07436063Phase 3Parkinson'sTerminated2541UPCR
NCT03193125Phase 3Cervical CaCompleted1190EDSS
Competitors (10)
DrugCompanyPhaseTargetMOA
RHH-7558RochePhase 1SGLT2Anti-Tau
NVS-4076NovartisPreclinicalTROP-2DLL3 ADC
NVS-5439NovartisPreclinicalBETAnti-Tau
NVS-8902NovartisPreclinicalTROP-2IL-13i
NVO-9630Novo NordiskPhase 2CD3Anti-Tau
ZanumavacamtenGSKPhase 2/3TROP-2BTKi
REG-2172RegeneronPhase 1/2PCSK9Anti-Tau
BGN-3305BeiGenePhase 2BCMAAnti-Tau
ION-1378IonisNDA/BLATROP-2RAS(ON)i
SovarasimodHalozymePhase 1/2WEE1Anti-Tau