← Pipeline|GRF-1969

GRF-1969

Phase 1/2
Source: Trial-derived·Trials: 2
Modality
Radioligand
MOA
ALKi
Target
KIF18A
Pathway
JAK/STAT
T2D
Development Pipeline
Preclinical
~Sep 2016
~Dec 2017
Phase 1
Mar 2018
Nov 2030
Phase 1Current
NCT08953427
2,353 pts·T2D
2018-032030-10·Not yet recruiting
NCT08649352
1,457 pts·T2D
2025-062030-11·Terminated
3,810 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (3)
2025-08-128mo agoEMA Filing· T2D
2030-10-244.6y awayPh2 Data· T2D
2030-11-254.7y awayPh2 Data· T2D
Trial Timeline
2018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q4
P1/2
Not yet…
P1/2
Termina…
Catalysts
EMA Filing
2025-08-12 · 8mo ago
T2D
Ph2 Data
2030-10-24 · 4.6y away
T2D
Ph2 Data
2030-11-25 · 4.7y away
T2D
TerminatedNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT08953427Phase 1/2T2DNot yet recr...2353OS
NCT08649352Phase 1/2T2DTerminated1457EFS
Competitors (10)
DrugCompanyPhaseTargetMOA
MiriosocimabPfizerPhase 1PARPALKi
NiranesiranJohnson & JohnsonPhase 2KIF18AEGFRi
MRK-7739Merck & CoPreclinicalIL-23ALKi
BMY-2495Bristol-Myers SquibbPhase 3KRASG12DALKi
DSN-5254Daiichi SankyoPhase 1B7-H3ALKi
SovacapivasertibAmgenPhase 3WEE1ALKi
ZanuratamabGilead SciencesPhase 1/2CDK2ALKi
GIL-2445Gilead SciencesPhase 2/3PSMAALKi
RiluinavolisibModernaNDA/BLAKIF18APLK4i
ALN-3284AlnylamPhase 2/3CDK2ALKi