← Pipeline|Gelicapivasertib

Gelicapivasertib

Approved
LUN-8561
Source: Trial-derived·Trials: 4
Modality
mRNA
MOA
IL-13i
Target
Pathway
Checkpoint
Epilepsy
Development Pipeline
Preclinical
~Feb 2016
~May 2017
Phase 1
~Aug 2017
~Nov 2018
Phase 2
~Feb 2019
~May 2020
Phase 3
~Aug 2020
~Nov 2021
NDA/BLA
~Feb 2022
~May 2023
Approved
Aug 2023
Mar 2029
ApprovedCurrent
NCT04950302
697 pts·Epilepsy
2024-092029-02·Terminated
NCT07721343
1,725 pts·Epilepsy
2025-092025-12·Active
NCT08755434
249 pts·Epilepsy
2023-082028-07·Terminated
+1 more trial
4,904 total pts1 indication
CompletedCurrentUpcoming
Catalysts (4)
2025-12-044mo agoPh3 Readout· Epilepsy
2028-07-132.3y awayPh3 Readout· Epilepsy
2029-02-012.8y awayPh3 Readout· Epilepsy
2029-03-062.9y awayPh3 Readout· Epilepsy
Trial Timeline
Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2
Approved
Termina…
Approved
Active
Approved
Termina…
Approved
Active
Catalysts
Ph3 Readout
2025-12-04 · 4mo ago
Epilepsy
Ph3 Readout
2028-07-13 · 2.3y away
Epilepsy
Ph3 Readout
2029-02-01 · 2.8y away
Epilepsy
Ph3 Readout
2029-03-06 · 2.9y away
Epilepsy
ActiveTerminated|StartCompletionToday
Trials (4)
NCTPhaseIndicationStatusNEP
NCT04950302ApprovedEpilepsyTerminated697EDSS
NCT07721343ApprovedEpilepsyActive1725PFS
NCT08755434ApprovedEpilepsyTerminated249PASI75
NCT04622127ApprovedEpilepsyActive2233LiverFat
Competitors (10)
DrugCompanyPhaseTargetMOA
PFE-7550PfizerPhase 3KIF18Ai
SotovorutinibPfizerApprovedCGRPant
VoxaderotideJohnson & JohnsonNDA/BLAPI3KαIL-13i
RHH-7975RochePhase 3FXIaIL-13i
NVS-8902NovartisPreclinicalTROP-2IL-13i
GozesotorasibBristol-Myers SquibbNDA/BLAHER2IL-13i
BemalucimabBristol-Myers SquibbPhase 1/2SGLT2i
BMY-4586Bristol-Myers SquibbPreclinicalKRASG12CIL-13i
DatobrutinibSanofiPhase 3HER2
DSN-791Daiichi SankyoNDA/BLAAuroraAi