← Pipeline|Kemazanubrutinib

Kemazanubrutinib

Phase 1/2
XER-7677
Source: Trial-derived·Trials: 2
Modality
ASO
MOA
STINGag
Target
TYK2
Pathway
T-cell
NarcolepsyRB
Development Pipeline
Preclinical
~Dec 2018
~Mar 2020
Phase 1
Jun 2020
Jun 2029
Phase 1Current
NCT07732855
1,425 pts·RB
2020-062029-06·Active
NCT04665613
1,527 pts·RB
2023-032026-11·Recruiting
2,952 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2026-11-248mo awayPh2 Data· RB
2029-06-213.2y awayPh2 Data· RB
Trial Timeline
Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3
P1/2
Active
P1/2
Recruit…
Catalysts
Ph2 Data
2026-11-24 · 8mo away
RB
Ph2 Data
2029-06-21 · 3.2y away
RB
RecruitingActive|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT07732855Phase 1/2RBActive1425DAS28
NCT04665613Phase 1/2RBRecruiting1527HAM-D
Competitors (10)
DrugCompanyPhaseTargetMOA
VoxacilimabPfizerPhase 2TYK2CAR-T BCMA
RHH-5389RochePreclinicalRETSTINGag
MRK-3732Merck & CoPhase 1TYK2PARPi
SNY-5894SanofiApprovedCFTRSTINGag
SNY-4496SanofiPhase 2/3CD3STINGag
SNY-5783SanofiPhase 1/2METSTINGag
DSN-1421Daiichi SankyoPhase 3Nectin-4STINGag
GIL-4361Gilead SciencesPreclinicalPCSK9STINGag
INC-5849IncytePhase 2PCSK9STINGag
MiritinibNeurocrinePhase 3TIGITSTINGag