← Pipeline|Kemavorutinib

Kemavorutinib

Approved
EXA-5914
Source: Trial-derived·Trials: 1
Modality
Radioligand
MOA
Menini
Target
JAK2
Pathway
Cell Cycle
SCD
Development Pipeline
Preclinical
~May 2017
~Aug 2018
Phase 1
~Nov 2018
~Feb 2020
Phase 2
~May 2020
~Aug 2021
Phase 3
~Nov 2021
~Feb 2023
NDA/BLA
~May 2023
~Aug 2024
Approved
Nov 2024
Oct 2025
ApprovedCurrent
NCT07161769
2,883 pts·SCD
2024-112025-10·Active
2,883 total pts1 indication
CompletedCurrentUpcoming
Catalysts (1)
2025-10-066mo agoPh3 Readout· SCD
Trial Timeline
2025Q2Q3Q4
Approved
Active
Catalysts
Ph3 Readout
2025-10-06 · 6mo ago
SCD
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT07161769ApprovedSCDActive2883BodyWt
Competitors (10)
DrugCompanyPhaseTargetMOA
MavutenlimabJohnson & JohnsonPhase 3Cl18.2Menini
IvorelsinEli LillyApprovedJAK1Menini
NVO-2974Novo NordiskNDA/BLAPARPMenini
GMA-5010GenmabPhase 3JAK2TROP-2 ADC
TeravorutinibIlluminaPhase 2JAK2PRMT5i
AXS-4984AxsomePreclinicalJAK2BiTE
CapirapivirTG TherapeuticsApprovedJAK2AuroraAi
OlpafutibatinibImmunocoreApprovedSMN2Menini
ZenorelsinDisc MedicineNDA/BLAJAK2CD47i
IRO-8712Disc MedicinePreclinicalJAK2EGFRi