← Pipeline|Rimavorutinib

Rimavorutinib

Phase 1
WIN-7623
Source: Trial-derived·Trials: 2
Modality
Gene Therapy
MOA
C5i
Target
RET
Pathway
NF-κB
OCD
Development Pipeline
Preclinical
~May 2023
~Aug 2024
Phase 1
Nov 2024
Feb 2030
Phase 1Current
NCT04357342
2,540 pts·OCD
2024-112028-05·Recruiting
NCT06851408
902 pts·OCD
2025-092030-02·Terminated
3,442 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2028-05-262.2y awayInterim· OCD
2030-02-053.9y awayInterim· OCD
Trial Timeline
Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030
P1
Recruit…
P1
Termina…
Catalysts
Interim
2028-05-26 · 2.2y away
OCD
Interim
2030-02-05 · 3.9y away
OCD
RecruitingTerminated|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT04357342Phase 1OCDRecruiting2540EASI-75
NCT06851408Phase 1OCDTerminated902ORR
Competitors (10)
DrugCompanyPhaseTargetMOA
RHH-5389RochePreclinicalRETSTINGag
FixanesiranAbbViePreclinicalRETJAK1/2i
BMY-8678Bristol-Myers SquibbApprovedRETMDM2i
DSN-2247Daiichi SankyoNDA/BLAEZH2C5i
VRT-1576Vertex PharmaPhase 2/3RETSHP2i
ARG-3458ArgenxPreclinicalRETIL-17i
RimabrutinibMadrigal PharmaPhase 1/2GPRC5DC5i
NidaratamabKrystal BiotechPreclinicalRETIL-17i
XEN-577Xenon PharmaPhase 2/3C5C5i
FixabrutinibVervePhase 1RETFcRni