← Pipeline|Olpasertib

Olpasertib

Phase 2
069-3718
Source: Trial-derived·Trials: 2
Modality
Gene Editing
MOA
VEGFi
Target
MALT1
Pathway
T-cell
RCCCRCRB
Development Pipeline
Preclinical
~Dec 2017
~Mar 2019
Phase 1
~Jun 2019
~Sep 2020
Phase 2
Dec 2020
Apr 2031
Phase 2Current
NCT06970066
1,647 pts·RB
2025-122031-04·Not yet recruiting
NCT08200124
1,200 pts·CRC
2020-12TBD·Recruiting
2,847 total pts2 indications
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2031-04-035.0y awayPh2 Data· RB
Trial Timeline
Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q42031Q2
P2
Recruit…
P2
Not yet…
Catalysts
Ph2 Data
2031-04-03 · 5.0y away
RB
RecruitingNot yet recruiting|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT06970066Phase 2RBNot yet recr...1647PASI75
NCT08200124Phase 2CRCRecruiting1200EFS
Competitors (10)
DrugCompanyPhaseTargetMOA
JNJ-8232Johnson & JohnsonNDA/BLAMALT1SGLT2i
MRK-5413Merck & CoPhase 1GLP-1RVEGFi
DoxasotorasibAbbViePhase 2CD38VEGFi
BMY-7975Bristol-Myers SquibbPhase 1MALT1WRNi
CeviderotideNovo NordiskPreclinicalIL-13VEGFi
GSK-6516GSKPhase 1/2MALT1PARPi
VRT-6833Vertex PharmaPreclinicalALKVEGFi
BII-5240BiogenPhase 2/3MALT1HPK1i
ALN-3958AlnylamPhase 2MALT1PARPi
CevisacituzumabAlnylamPreclinicalMALT1SOS1i