← Pipeline|Mavuzanubrutinib

Mavuzanubrutinib

Phase 1/2
MGT-3302
Source: Trial-derived·Trials: 1
Modality
ERT
MOA
PRMT5i
Target
IL-17A
Pathway
Checkpoint
MCLCTCLAS
Development Pipeline
Preclinical
~Dec 2020
~Mar 2022
Phase 1
Jun 2022
Jul 2025
Phase 1Current
NCT07440100
975 pts·CTCL
2022-062025-07·Active
975 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2025-07-109mo agoPh2 Data· CTCL
Trial Timeline
Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3
P1/2
Active
Catalysts
Ph2 Data
2025-07-10 · 9mo ago
CTCL
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT07440100Phase 1/2CTCLActive975CR
Competitors (10)
DrugCompanyPhaseTargetMOA
LLY-6079Eli LillyPhase 2MDM2PRMT5i
RHH-8550RocheApprovedBCL-2PRMT5i
RHH-682RochePhase 2FXIaPRMT5i
GeliderotideNovartisNDA/BLAIL-17ABCL-2i
TalainavolisibNovo NordiskPreclinicalKRASG12DPRMT5i
TirasotorasibTakedaNDA/BLAIL-17ACDK2i
AMG-4531AmgenPhase 2/3KRASG12CPRMT5i
GIL-9779Gilead SciencesPhase 1IL-17ABCMA ADC
GIL-9142Gilead SciencesPhase 1FXIaPRMT5i
SemainavolisibGilead SciencesPhase 2PARPPRMT5i