← Pipeline|255-7731

255-7731

Phase 1
Source: Trial-derived·Trials: 1
Modality
Peptide
MOA
MDM2i
Target
EZH2
Pathway
PI3K/AKT
RBWilmsMM
Development Pipeline
Preclinical
~Feb 2022
~May 2023
Phase 1
Aug 2023
Phase 1Current
NCT08481446
1,314 pts·Wilms
2023-08TBD·Recruiting
1,314 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2025-12-273mo agoOrphan Drug· Wilms
Trial Timeline
Q42024Q2Q3Q42025Q2Q3Q4
P1
Recruit…
Catalysts
Orphan Drug
2025-12-27 · 3mo ago
Wilms
Recruiting|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT08481446Phase 1WilmsRecruiting1314NT-proBNP
Competitors (10)
DrugCompanyPhaseTargetMOA
DoxacapivasertibEli LillyPhase 3APOC3MDM2i
BMY-8678Bristol-Myers SquibbApprovedRETMDM2i
DSN-2247Daiichi SankyoNDA/BLAEZH2C5i
AMG-415AmgenPhase 1CDK2MDM2i
GIL-2037Gilead SciencesApprovedKRASG12DMDM2i
CapiglumideBioNTechPreclinicalCGRPMDM2i
HAL-9635HalozymePhase 2/3EZH2Cl18.2
RimasertibExelixisPhase 3B7-H3MDM2i
180-6098Innovent BioPhase 1ALKMDM2i
ElralucimabAxsomePhase 2CDK4/6MDM2i