← Pipeline|Zanumavacamten

Zanumavacamten

Phase 2/3
GSK-5385
By GSK
Source: Trial-derived·Trials: 1
Modality
Cell Therapy
MOA
BTKi
Target
TROP-2
Pathway
Angiogenesis
MDSADHDRA
Development Pipeline
Preclinical
~Aug 2016
~Nov 2017
Phase 1
~Feb 2018
~May 2019
Phase 2
Aug 2019
Jun 2029
Phase 2Current
NCT03480272
389 pts·MDS
2019-082029-06·Terminated
389 total pts1 indication
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2029-06-253.2y awayPh3 Readout· MDS
Trial Timeline
Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3
P2/3
Termina…
Catalysts
Ph3 Readout
2029-06-25 · 3.2y away
MDS
Terminated|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT03480272Phase 2/3MDSTerminated389UPCR
Competitors (10)
DrugCompanyPhaseTargetMOA
NVS-4076NovartisPreclinicalTROP-2DLL3 ADC
NVS-8902NovartisPreclinicalTROP-2IL-13i
AZN-8281AstraZenecaPhase 1SHP2BTKi
BMY-3371Bristol-Myers SquibbPhase 3WRNBTKi
NVO-7872Novo NordiskNDA/BLAB7-H3BTKi
NVO-6275Novo NordiskPhase 1SMN2BTKi
TAK-2403TakedaPhase 2WEE1BTKi
LisorapivirTakedaPreclinicalWRNBTKi
IvosotorasibVertex PharmaPreclinicalCD38BTKi
MRN-8133ModernaPhase 2PD-1BTKi