← Pipeline|Motarapivir

Motarapivir

Preclinical
GSK-6551
By GSK
Source: Trial-derived·Trials: 2
Modality
Multispecific
MOA
IL-23i
Target
AuroraA
Pathway
Cell Cycle
ALLHeart Failure
Development Pipeline
Preclinical
Oct 2017
Aug 2030
PreclinicalCurrent
NCT07268818
2,747 pts·Heart Failure
2017-102028-04·Terminated
NCT04024918
280 pts·Heart Failure
2019-012030-08·Completed
3,027 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2028-04-042.0y awayInterim· Heart Failure
2030-08-254.4y awayInterim· Heart Failure
Trial Timeline
Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q4
Preclinical
Termina…
Preclinical
Complet…
Catalysts
Interim
2028-04-04 · 2.0y away
Heart Failure
Interim
2030-08-25 · 4.4y away
Heart Failure
CompletedTerminated|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT07268818PreclinicalHeart FailureTerminated2747Biomarker
NCT04024918PreclinicalHeart FailureCompleted280Biomarker
Competitors (10)
DrugCompanyPhaseTargetMOA
GSK-6983GSKPhase 2ALKIL-23i
BAY-8733BayerPreclinicalAuroraABETi
ZenotapinarofVertex PharmaPreclinicalCD38IL-23i
BNT-8090BioNTechPhase 2AuroraAPD-L1i
ARG-6988ArgenxPreclinicalAuroraACDK2i
BemasotorasibExelixisPhase 2CD38IL-23i
TirasotorasibViking TherapeuticsPhase 1CFTRIL-23i
SemamavacamtenIdeaya BioPhase 1/2AuroraABTKi
CevinaritidePraxis PrecisionPhase 3AuroraAFcRni
SND-4562SyndaxNDA/BLAAuroraACAR-T CD19