← Pipeline|APT-1263

APT-1263

Phase 1
Source: Trial-derived·Trials: 1
Modality
Radioligand
MOA
CGRPant
Target
VEGF
Pathway
Amyloid
LN
Development Pipeline
Preclinical
~Jan 2023
~Apr 2024
Phase 1
Jul 2024
Nov 2030
Phase 1Current
NCT04034490
2,540 pts·LN
2024-072030-11·Active
2,540 total pts1 indication
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (1)
2030-11-254.7y awayInterim· LN
Trial Timeline
Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q42030Q2Q3Q4
P1
Active
Catalysts
Interim
2030-11-25 · 4.7y away
LN
Active|StartCompletionToday
Trials (1)
NCTPhaseIndicationStatusNEP
NCT04034490Phase 1LNActive2540HbA1c
Competitors (10)
DrugCompanyPhaseTargetMOA
TerafutibatinibPfizerPhase 1/2CD38CGRPant
SotovorutinibPfizerApprovedCGRPant
ZanuderotideNovartisPhase 1/2VEGFCD3xCD20
ABB-3060AbbViePhase 2LAG-3CGRPant
TAK-8730TakedaPhase 2VEGFFXIai
GIL-2011Gilead SciencesPreclinicalVEGFSOS1i
GIL-6239Gilead SciencesPhase 2TNFαCGRPant
BemazumabRegeneronPhase 1VEGFTROP-2 ADC
TezecilimabRegeneronApprovedIL-23CGRPant
INC-2432IncytePhase 2CD47CGRPant