← Pipeline|Mavuinavolisib

Mavuinavolisib

Preclinical
RNA-543
Source: Trial-derived·Trials: 2
Modality
Gene Therapy
MOA
Cl18.2
Target
VEGF
Pathway
PD-1/PD-L1
CSUGBM
Development Pipeline
Preclinical
Jun 2017
Sep 2029
PreclinicalCurrent
NCT07018356
666 pts·CSU
2019-052029-08·Completed
NCT07645707
734 pts·CSU
2017-062029-09·Completed
1,400 total pts1 indication
Phase 1
Phase 2
Phase 3
NDA/BLA
Approved
CompletedCurrentUpcoming
Catalysts (2)
2029-08-133.4y awayInterim· CSU
2029-09-223.5y awayInterim· CSU
Trial Timeline
Q2Q3Q42018Q2Q3Q42019Q2Q3Q42020Q2Q3Q42021Q2Q3Q42022Q2Q3Q42023Q2Q3Q42024Q2Q3Q42025Q2Q3Q42026Q2Q3Q42027Q2Q3Q42028Q2Q3Q42029Q2Q3Q4
Preclinical
Complet…
Preclinical
Complet…
Catalysts
Interim
2029-08-13 · 3.4y away
CSU
Interim
2029-09-22 · 3.5y away
CSU
Completed|StartCompletionToday
Trials (2)
NCTPhaseIndicationStatusNEP
NCT07018356PreclinicalCSUCompleted666EASI-75
NCT07645707PreclinicalCSUCompleted734SeizFreq
Competitors (10)
DrugCompanyPhaseTargetMOA
ZanuderotideNovartisPhase 1/2VEGFCD3xCD20
ZorivorutinibBristol-Myers SquibbApprovedDLL3Cl18.2
TAK-8730TakedaPhase 2VEGFFXIai
GIL-2011Gilead SciencesPreclinicalVEGFSOS1i
BemazumabRegeneronPhase 1VEGFTROP-2 ADC
ElrarapivirRegeneronPhase 1GIP-RCl18.2
PemicapivasertibLegend BiotechPhase 3VEGFCDK4/6i
SematapinarofLegend BiotechNDA/BLAVEGFCGRPant
LEG-6533Legend BiotechNDA/BLAVEGFPARPi
HAL-9635HalozymePhase 2/3EZH2Cl18.2